Home / Articles / Heterocyclisation of trisubstituted formamidines containing an aryl or hetaryl substituent at the imine nitrogen atom

Heterocyclisation of trisubstituted formamidines containing an aryl or hetaryl substituent at the imine nitrogen atom

Gennady Veniaminovich Oshovsky 1
Gennady Veniaminovich Oshovsky
, 
Alexander Mikhailovich Pinchuk 1
Alexander Mikhailovich Pinchuk
1 Institute of Organic Chemistry, National Academy of Sciences of Ukraine, Kyiv
Published 30 November 1999
Communication , Volume 69, Issue 10, 845-860
6
Share
Cite this
GOST
 | 
Cite this
GOST
Oshovsky G. V., Pinchuk A. M. Heterocyclisation of trisubstituted formamidines containing an aryl or hetaryl substituent at the imine nitrogen atom // Russian Chemical Reviews. 2000. Vol. 69. No. 10. pp. 845-860.
GOST all authors (up to 50)
Oshovsky G. V., Pinchuk A. M. Heterocyclisation of trisubstituted formamidines containing an aryl or hetaryl substituent at the imine nitrogen atom // Russian Chemical Reviews. 2000. Vol. 69. No. 10. pp. 845-860.
RIS
 | 
Cite this
RIS
TY - JOUR
DO - 10.1070/RC2000v069n10ABEH000600
UR - https://rcr.colab.ws/publications/10.1070/RC2000v069n10ABEH000600
TI - Heterocyclisation of trisubstituted formamidines containing an aryl or hetaryl substituent at the imine nitrogen atom
T2 - Russian Chemical Reviews
AU - Oshovsky, Gennady Veniaminovich
AU - Pinchuk, Alexander Mikhailovich
PY - 2000
DA - 1999/11/30
PB - ANO Editorial Board of the journal Uspekhi Khimii
SP - 845-860
IS - 10
VL - 69
ER -
BibTex
 | 
Cite this
BibTex (up to 50 authors)
@article{2000_Oshovsky,
author = {Gennady Veniaminovich Oshovsky and Alexander Mikhailovich Pinchuk},
title = {Heterocyclisation of trisubstituted formamidines containing an aryl or hetaryl substituent at the imine nitrogen atom},
journal = {Russian Chemical Reviews},
year = {2000},
volume = {69},
publisher = {ANO Editorial Board of the journal Uspekhi Khimii},
month = {Nov},
url = {https://rcr.colab.ws/publications/10.1070/RC2000v069n10ABEH000600},
number = {10},
pages = {845--860},
doi = {10.1070/RC2000v069n10ABEH000600}
}
MLA
Cite this
MLA
Oshovsky, Gennady Veniaminovich, and Alexander Mikhailovich Pinchuk. “Heterocyclisation of trisubstituted formamidines containing an aryl or hetaryl substituent at the imine nitrogen atom.” Russian Chemical Reviews, vol. 69, no. 10, Nov. 2000, pp. 845-860. https://rcr.colab.ws/publications/10.1070/RC2000v069n10ABEH000600.
Views / Visits / Downloads
14 / 14 / 2

Abstract

Published data on the cyclisation of N1,N1-disubstituted N2-aryl- and N2-hetaryl-formamidines are analysed, described systematically and generalised. The bibliography includes 147 references.

References

1.
Reactions and synthetic uses of amidines
Boyd G.V.
Chemistry of Functional Groups , 1991
3.
Advances in the Chemistry of Amidines
Granik V.G.
Russian Chemical Reviews , 1983
4.
5
A. A. Krasnovskii
Dokl. Akad. Nauk SSSR , 1953
5.
6
V. B. Evstigneev
Dokl. Akad. Nauk SSSR , 1953
6.
7
E. Rabinowitch
"Photosynthesis" , 1956
7.
8
V. N. Kondrat'ev
"Kinetika Reaktsii v Gazovoi Faze" (Kinetics of Reactions in the Gas Phase) , 1959
8.
The reaction of benzyne with imines
Fishwick C.W., Gupta R.C., Storr R.C.
Journal of the Chemical Society Perkin Transactions 1 , 1984
9.
10
T. A. Kryukova
"Polyaro-graficheskii Analiz" (Polarographic Analysis) , 1959
10.
11
T. T. Bannister
Diss. Abstr. , 1959
13.
1-Amino-2-azadienes from the thermolysis of 2-amino-1-azirines. New reagents for the construction of pyridine and dihydropyridine rings
Demoulin A., Gorissen H., Hesbain-Frisque A.M., Ghosez L.
Journal of the American Chemical Society , 1975
15.
First Diels-Alder Reaction of Pyrazolyl Imines under Microwave Irradiation
Díaz-Ortiz A., Carrillo J.R., Gómez-Escalonilla M.J., de la Hoz A., Moreno A., Prieto P.
Synlett , 1998
18.
Addition reactions of heterocumulenes. III. Reaction of diketene with formamidine derivatives.
SAKAMOTO M., MIYAZAWA K., TOMIMATSU Y.
Chemical and Pharmaceutical Bulletin , 2011
22.
Cycloaddition reactions of isocyanates. Reaction of aryl isocyanates with N,N-dimethylformamide
Ulrich H., Tucker B., Stuber F.A., Sayigh A.A.
Journal of Organic Chemistry , 1968
24.
Reactions of aryl isocyanates with substituted formamides and formamidines
Dyer E., Majewski T.E., Travis J.D.
Journal of Organic Chemistry , 1968
25.
Synthesis of heterocyclic compounds. Part 34. Reactions of chlorosulphonyl isocyanate with carbon–nitrogen double bonds
Suschitzky H., Walrond R.E., Hull R.
Journal of the Chemical Society Perkin Transactions 1 , 1977
26.
27
A. A. Krasnovskii
Biofizika , 1956
27.
28
A. A. Krasnovskii
Dokl. Akad. Nauk SSSR , 1955
28.
Formation of [2 + 2] cycloadducts from heterocyclic formamidines and phenyl isocyanate
Tišbler M., Stanovnik B.
Journal of the Chemical Society Chemical Communications , 1980
32.
Isomerisation about the C–N and CN bonds of E- and Z-amidines
Hegarty A.F., Chandler A.
Journal of the Chemical Society Chemical Communications , 1980
33.
Unequivocal synthesis of 6-arylpteridines by intramolecular cycloaddition of azahexatrienes
Yoneda F., Higuchi M.
Journal of the Chemical Society Perkin Transactions 1 , 1977
37.
A novel synthesis of 8-arylaminotheophyllines
Senga K., Ichiba M., Kanazawa H., Nishigaki S., Higuchi M., Yoneda F.
Journal of Heterocyclic Chemistry , 1978
38.
A New Synthesis of Disubstituted 8-Aminopurine Derivatives
YONEDA F., HIGUCHI M., HAYAKAWA A.
Synthesis , 1975
39.
40
A. A. Krasnovskii
Biofizika , 1960
40.
41
A. A. Krasnovskii
Dokl. Akad. Nauk SSSR , 1950
41.
42
L. K. Obukhova
Izv. Akad. Nauk SSSR, Otd. Khim. Nauk , 1960
42.
43
N. Bunge
Ber. Deutsch. Chem. Ges. , 1870
43.
Pyrimidine derivatives and related compounds. XL. Synthesis of 7-substituted pyrimido(5,4-d)pyrimidines.
HIROTA K., YAMADA Y., ASAO T., KITADE Y., SENDA S.
Chemical and Pharmaceutical Bulletin , 2011
46.
47
G. Oster
"Research in Photosynthesis" , 1957
47.
48
A. A. Krasnovskii
Dokl. Akad. Nauk SSSR , 1955
50.
51
A. A. Krasnovskii
Dokl. Akad. Nauk SSSR , 1954
51.
52
V. B. Evstigneev
Dokl. Akad. Nauk SSSR , 1957
52.
53
D. Porretand E. Rabinowitch
Nature , 1937
53.
54
R. Livingston
J. Phys. Chem. , 1941
54.
55
G. A. Bogdanovskii
1958
55.
56
T. Iasui
Bull. Chem. Soc. Japan. , 1935
56.
57
R. Livingston
"Research in Photosynthesis" , 1957
57.
58
N. E. Khomutov
1953
58.
59
H. Linshitz
"Research in Photosynthesis" , 1957
59.
60
A. N. Terenin
Optika i Spektrosk. , 1956
60.
61
A. N. Terenin
1959
61.
62
A. A. Krasnovskii
"Sbornik, Voprosy Khimicheskoi Kinetiki" (Symposium, Problems of Chemical Kinetics) , 1955
62.
63
1930
63.
64
Chem. Zentr. II , 1931
64.
65
A. A. Krasnovskii
Biofizika , 1959
65.
66
V. B. Evstigneev
Dokl. Akad. Nauk SSSR , 1950
66.
67
N. N. Mel'nikov
Zhur. Obshch. Khim. , 1940
67.
68
N. N. Mel'nikov
Zhur. Obshch. Khim. , 1946
68.
69
B. Commoner
1958
69.
70
N. Bubnov
Biofizika , 1960
70.
71
Yu. A. Shlyapnikov
Vysokomol. Soed. , 1962
71.
Cushingʼs Disease—18 Yearsʼ Experience
URBANIC R.C., GEORGE J.M.
Medicine (United States) , 2006
72.
73
T. Skwarski
Chem. Abs. , 1957
73.
74
F. F. Litvin
Uspekhi Fiz. Nauk , 1960
74.
75
V. B. Evstigneev
Dokl. Akad. Nauk SSSR , 1950
75.
76
A. N. Terenin
"Fotokhimiya Krasitelei" (The Photochemistry of Dyes) , 1947
76.
77
A. A. Krasnovskii
Dokl. Akad. Nauk SSSR , 1948
77.
78
A. A. Krasnovskii
Dokl. Akad. Nauk SSSR , 1949
78.
79
A. A. Krasnovskii
Dokl. Akad. Nauk SSSR , 1952
79.
80
N. N. Mel'nikov
Zhur. Obshch. Khim. , 1937
80.
81
J. C. Ghosh
J. Indian Chem. Soc. , 1934
81.
The Synthetic Potentialities of Nitriles in Heterocyclic Synthesis
Mourad Sherif S., Hilmy Elnagdi M., Milad Mohareb R.
Heterocycles , 1987
82.
83
A. A. Krasnovskii
Dokl. Akad. Nauk SSSR , 1947
83.
84
A. A. Krasnovskii
Dokl. Akad. Nauk SSSR , 1947
85.
86
V. B. Evstigneev
Dokl. Akad. Nauk SSSR , 1958
86.
87
J. F. Arens
"Advances in Organic Chemistry" , 1960
87.
88
A. A. Krasnovskii
Dokl. Akad. Nauk SSSR , 1946
88.
89
A. A. Krasnovskii
Izd. Akad. Nauk SSSR, Moscow , 1955
89.
90
V. B. Evstigneev
Dokl. Akad. Nauk SSSR , 1951
90.
91
L. M. Vorob'eva
Biokhimiya , 1956
91.
92
A. A. Krasnovskii
Dokl. Akad. Nauk SSSR , 1948
92.
93
V. B. Evstigneev
Dokl. Akad. Nauk SSSR , 1956
93.
Use of a Pharmacophore Model for the Design of EGF-R Tyrosine Kinase Inhibitors:  4-(Phenylamino)pyrazolo[3,4-d]pyrimidines
Traxler P., Bold G., Frei J., Lang M., Lydon N., Mett H., Buchdunger E., Meyer T., Mueller M., Furet P.
Journal of Medicinal Chemistry , 1997
95.
96
L. M. Vorob'eva
Biokhimiya , 1958
96.
97
A. N. Terenin
Dokl. Akad. Nauk SSSR , 1952
97.
98
W. Franke
Chem. Zentr. , 1954
98.
99
V. V. Zolotarev
1938
99.
100
V. V. Zolotarev
Chem. Abs. , 1941
100.
101
M. F. Shostakovskii
Izv. Akad. Nauk SSSR, Otd. Khim. Nauk , 1960
101.
102
F. Fichter
Helv. Chim. Acta , 1922
103.
104
O. P. Osipova
Dokl. Akad. Nauk SSSR , 1950
104.
105
F. F. Litvin
Dokl. Akad. Nauk SSSR , 1958
105.
106
F. Fichter
Helv. Chim. Acta , 1927
108.
109
F. Ficher
Bull. Soc. chim. France (4) , 1916
109.
110
M. F. Shostakovskii
Dokl. Akad. Nauk SSSR , 1960
110.
111
M. Calvin
1956
111.
112
A. G. Pozdeeva
Zhur. Prikl. Khim. , 1952
112.
113
H. Blum
"Photodynamic Action and Diseases caused Light" , 1940
113.
114
L. Segal
"Chemical Reactions of Polymers" , 1964
114.
115
A. A. Krasnovskii
Dokl. Akad. Nauk SSSR , 1957
115.
116
V. B. Evstigneev
Dokl. Akad. Nauk SSSR , 1957
116.
Pyridazines.LIX. Synthesis ofc-annelated pyridazines from 3-amino-4-pyridazinecarbonitrile
Haider N., Heinisch G., Wanko R.
Journal of Heterocyclic Chemistry , 1991
118.
119
V. V. Levchenko
Zhur. Obshch. Khim. , 1947
119.
120
V. V. Levchenko
Zhur. Obshch. Khim. , 1948
120.
121
V. V. Korshak
Izv. Akad. Nauk SSSR, Otd. Khim. Nauk , 1953
121.
122
S. R. Rafikov
Izv. Akad. Nauk SSSR, Otd. Khim. Nauk , 1953
122.
123
V. V. Levchenko
Zhur. Obshch. Khim. , 1952
123.
124
V. V. Levchenko
Zhur. Obshch. Khim. , 1952
124.
Heterocycles. VII. Novel and Facile Syntheses of s-Triazolo-[4, 3-a] [1, 4] benzodiazepine Derivatives
125.
Some New Synthetic Approaches for the Preparation of Pteridine-3-oxides and Pteridines
Kočevar M., Kocevar M., Stanovnik B., Tisler M.
Heterocycles , 1981
126.
Syntheses and transformations of some 1,2,4-oxadiazolylpyrazines
Kočevar M., Stanovnik B., Tišler M.
Journal of Heterocyclic Chemistry , 1982
127.
128
J. Wiemann
Bull. Soc. chim. France , 1952
128.
129
J. Wiemann
Bull. Soc. chim. France , 1955
129.
Synthesis and central nervous system stimulant activity of camphor-1,2,4-benzotriazines fused with five and six-membered heterocycles
Nagai S., Ueda T., Takamura M., Nagatsu A., Murakami N., Sakakibara J.
Journal of Heterocyclic Chemistry , 1998
130.
131
N. Thooi
Compt. rend. , 1958
131.
An unequivocal synthesis of some substituted 1,2,4-triazolo[1,5-a]pyrimidines
Stanovnik B., Urleb U., Tišler M.
Monatshefte fur Chemie , 1987
132.
Heterocycles. CXVIII. Pyridazines. LXVI. Novel method of annelation of the 1,2,4-triazole ring of the N2-C3 bond to azines
136.
Potential antisecretory antidiarrheals. 2. .alpha.2-Adrenergic 2-[(aryloxy)alkyl]imidazolines
Moormann A.E., Pitzele B.S., Jones P.H., Gullikson G.W., Albin D., Yu S.S., Bianchi R.G., Sanguinetti E.L., Rubin B.
Journal of Medicinal Chemistry , 1990
137.
New quinoxaline and pyrimido[4,5-b]quinoxaline derivatives. Potential antihypertensive and blood platelet antiaggregating agents
138.
A New Indole Synthesis1
Lorenz R.R., Tullar B.F., Koelsch C.F., Archer S.
Journal of Organic Chemistry , 1965
140.
141
Friedl.
141.
Formation of indoles and quinolines by flash vacuum pyrolysis
142.
4,7-Diazaindole Derivatives
Klutchko S., Hansen H.V., Meltzer R.I.
Journal of Organic Chemistry , 1965
143.
144
1912
144.
145
Friedl.
145.
146
V. V. Korshak
Dokl. Akad. Nauk SSSR , 1952
146.
147
Y. Sasada
Acta Cryst. , 1898
147.
Synthesis of (aryloxy)alkylamines. 2. Novel imidazo-fused heterocycles with calcium channel blocking and local anesthetic activity
Sanfilippo P.J., Urbanski M., Press J.B., Dubinsky B., Moore J.B.
Journal of Medicinal Chemistry , 1988
148.
149
V. V. Korshak
Dokl. Akad. Nauk SSSR , 1954
149.
150
Ya. E. Bernadskaya
"Iskusstvennoe Volokno" (Artificial Fibres) , 1952
151.
152
W. Albert
Trans. Electrochem. Soc. , 1943
153.
154
Friedl.
154.
155
M. V. Mal'tsev
Izv. Vys. Ucheb. Zaved., Tsvet. Met. , 1960
155.
156
J. S. Fruton
J. Biol. Med. , 1950
156.
Addition of nitroalkanes to -halo-nitrobenzenes
Reid J.G., Reny Runge J.H.
Tetrahedron Letters , 1990
157.
158
Friedl.
159.
160
1912
160.
161
Friedl.
161.
162
1917
162.
163
Friedl.
164.
Synthesis and transformations of some pyrido[2,3-d]pyrimidines
Kočevar M., Koller J., Stanovnik B., Tišler M.
Monatshefte fur Chemie , 1987
165.
166
1917
166.
167
Friedl.
168.
169
Friedl.
169.
170
1918
171.
172
1918
172.
173
Friedl.
173.
The transformations of 4-heteroarylaminomethylene-5(4H)-oxazolones into dehydropeptide derivatives
Aljaẑ-Roẑiĉ M., Svete J., Stanovnik B.
Journal of Heterocyclic Chemistry , 1995
175.
Transformation of Amines and N-Heteroarylformamidines into Esters of Substituted b-Amino-a,b-dehydro-a-amino Acids
176.
The synthesis of β-heteroarylamino-α,β-dehydro-α-amino acid and β-heteroarylamino-α-amino acid derivatives
Svete J., Stanovnik B., Tišler M., Golič L., Leban I.
Journal of Heterocyclic Chemistry , 1989
177.
178
1946
178.
New Synthetic Approach for Azolopurines and Analogs
Tisler M., Stanovnik B., Zrimsek Z.
Heterocycles , 1982
179.
180
1946
180.
New synthesis of 5H-pyrrolo[3,2-d]pyrimidines via pyrimido[5,4-c]pyridazines
Klein R.S., Lim M., Tam S.Y., Fox J.J.
Journal of Organic Chemistry , 1978
183.
Functionalized Enamines in the Synthesis of Some Heterocyclic Compounds
Tisler M., Golic L., Stropnik C., Stanovnic B.
Heterocycles , 1987
184.
185
1954
185.
186
Chem. Abs. , 1956
186.
187
1954
187.
188
Chem. Abs. , 1955
188.
189
M. Godchot
Bull. Soc. chim. France (5) , 1913
189.
190
H. Law
J. Chem. Soc. , 1912